SCHEMBL6589548

SCHEMBL6589548

COc1nsnc1N1CCN(CC(Cc2ccccc2)N(C)C(=O)N2CCOCC2)CC1

nearest known ligand 0.74

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.74
ALDH1A1 P00352 6/20 0.46
TSHR P16473 2/20 0.46
ALOX15 P16050 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MAPK1 P28482 1/20 0.46
KMT2A Q03164 3/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
LMNA P02545 1/20 0.44
MAPT P10636 2/20 0.44
POLB P06746 1/20 0.44
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
LIPA P38571 4/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589369 0.88 HTR1A (0.72) HTR1AALDH1A1TSHRALOX15HSD17B10
SCHEMBL6588749 0.85 HTR1A (1.00) HTR1AALDH1A1TSHRALOX15HSD17B10
SCHEMBL6588614 0.76 HTR1A (0.66) HTR1AALDH1A1TSHRALOX15HSD17B10
SCHEMBL6586728 0.76 HTR1A (0.66) HTR1AALDH1A1TSHRALOX15HSD17B10
SCHEMBL6586733 0.73 HTR1A (0.61) HTR1AALDH1A1TSHRALOX15HSD17B10
SCHEMBL6588617 0.73 HTR1A (0.61) HTR1AALDH1A1TSHRALOX15HSD17B10
SCHEMBL6586789 0.65 HTR1A (0.61) HTR1AALDH1A1TSHRALOX15HSD17B10
Hydrochloric Acid SCHEMBL4728303 0.63 ALDH1A1 (0.50) ALDH1A1HSD17B10MAPK1KMT2ALMNA
SCHEMBL31703718 0.62 KMT2A (0.57) ALDH1A1TSHRALOX15HSD17B10KMT2A
SCHEMBL9800484 0.62 KMT2A (0.59) ALDH1A1TSHRALOX15HSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002538152-A 2002-11-12 JP claimed
EP-1161424-A1 NEW DIAZOLE DERIVATIVES AS SEROTONERGIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 2001-12-12 EP claimed
WO-2000051999-A1 NEW DIAZOLE DERIVATIVES AS SEROTONERGIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-09-08 WO claimed
EP-1161424-B1 NEW DIAZOLE DERIVATIVES AS SEROTONERGIC AGENTS WYETH CORP (US) 2004-06-02 EP disclosed