SCHEMBL6603919

SCHEMBL6603919

CC(C)OC(=O)CCN1CCN(CC2CN(c3ccc(C(=N)NC(=O)c4ccc5ccccc5c4)cc3)C(=O)O2)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
SIGMAR1 Q99720 8/20 0.41
POLB P06746 1/20 0.40
HTR1A P08908 6/20 0.40
SLC6A4 P31645 2/20 0.39
SLC6A2 P23975 1/20 0.39
F10 P00742 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602415 0.93 ITGB3 (0.48) ITGB3ITGA2BSIGMAR1HTR1AF10
SCHEMBL6601180 0.93 ITGB3 (0.45) ITGB3ITGA2BSIGMAR1POLBHTR1A
SCHEMBL6606831 0.92 ITGB3 (0.44) ITGB3ITGA2BSIGMAR1F10
SCHEMBL6605691 0.90 ITGB3 (0.51) ITGB3ITGA2BSIGMAR1POLBHTR1A
SCHEMBL6602885 0.90 ITGB3 (0.42) ITGB3ITGA2BSIGMAR1POLBHTR1A
SCHEMBL6600977 0.89 ALDH1A1 (0.43) ITGB3ITGA2BSIGMAR1F10
SCHEMBL7314871 0.89 HTR1A (0.44) ITGB3ITGA2BSIGMAR1POLBHTR1A
SCHEMBL6603912 0.88 ITGB3 (0.43) ITGB3ITGA2BSIGMAR1
SCHEMBL6600922 0.88 SIGMAR1 (0.44) ITGB3ITGA2BSIGMAR1
SCHEMBL6601430 0.88 ITGB3 (0.43) ITGB3ITGA2BSIGMAR1POLBHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed