SCHEMBL6603974

SCHEMBL6603974

Cc1ccccc1CC1=C(O)CC(CCc2ccccc2)(c2ccccc2)OC1=O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
LDHA P00338 2/20 0.36
CNR2 P34972 3/20 0.34
GPR55 Q9Y2T6 2/20 0.34
CNR1 P21554 1/20 0.34
EGFR P00533 1/20 0.34
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 2/20 0.33
FFAR1 O14842 1/20 0.33
HTT P42858 1/20 0.33
OPRM1 P35372 2/20 0.33
OPRL1 P41146 2/20 0.33
MAPT P10636 1/20 0.33
ASAH1 Q13510 1/20 0.32
KDM4E B2RXH2 2/20 0.32
UTS2R Q9UKP6 1/20 0.32
DAO P14920 1/20 0.32
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026445 0.91 ALDH1A1 (0.38) ALDH1A1LDHAEGFRGAAL3MBTL1
SCHEMBL6603192 0.88 LDHA (0.39) LDHAEGFRGAAL3MBTL1LMNA
SCHEMBL6609678 0.87 LDHA (0.40) LDHAEGFRGAAL3MBTL1OPRM1
SCHEMBL8658523 0.86 TAAR1 (0.41) ALDH1A1LDHACNR2CNR1GAA
SCHEMBL6602958 0.86 LDHA (0.38) LDHACNR2GPR55EGFRFFAR1
SCHEMBL6603612 0.84 OPRM1 (0.38) ALDH1A1LDHACNR1EGFRGAA
SCHEMBL6608780 0.83 NPC1 (0.36) ALDH1A1LDHAL3MBTL1LMNAASAH1
SCHEMBL6608872 0.83 LDHA (0.41) LDHAEGFRGAAL3MBTL1LMNA
SCHEMBL6603481 0.82 ASAH1 (0.34) LDHACNR2GPR55HTTMAPT
SCHEMBL6604120 0.81 OPRK1 (0.37) LDHAEGFROPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142887-B1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents PARKE DAVIS & CO (US) 2004-04-07 EP disclosed
EP-1142887-A1 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents PARKE, DAVIS & COMPANY (US) 2001-10-10 EP disclosed
US-5936128-A BENZENETHIOL COMPOUNDS AS INTERMEDIATES; BACTERICIDES, VIRICIDES; HIV WARNER-LAMBERT COMPANY (US) 1999-08-10 US disclosed
US-5840751-A ADMINISTERING IN THE TREATMENT OF INFECTION OR DISEASE CAUSED BY A RETROVIRUS WARNER-LAMBERT COMPANY (US) 1998-11-24 US disclosed
US-5789440-A 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents WARNER-LAMBERT COMPANY (US) 1998-08-04 US disclosed
EP-0729464-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014012-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014011-A2 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed