SCHEMBL6612337

SCHEMBL6612337

O=C1CNC(=O)C2(CCN(CCc3ccccc3)CC2)N1CC(c1ccccc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.48
CYP2D6 P10635 2/20 0.48
CHRM2 P08172 1/20 0.48
ADRA2A P08913 1/20 0.48
TSHR P16473 1/20 0.48
DRD1 P21728 1/20 0.48
MAPT P10636 2/20 0.47
KMT2A Q03164 2/20 0.47
SIGMAR1 Q99720 4/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
OPRM1 P35372 3/20 0.42
OPRD1 P41143 2/20 0.42
OPRK1 P41145 2/20 0.42
OPRL1 P41146 2/20 0.42
CCR5 P51681 5/20 0.42
HTR2A P28223 3/20 0.41
HTR2C P28335 3/20 0.41
HTR2B P41595 3/20 0.41
DRD2 P14416 2/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6614708 0.93 CCR5 (0.47) LMNACYP2D6TSHRMAPTKMT2A
SCHEMBL6613155 0.92 CCR5 (0.51) LMNACYP2D6MAPTKMT2ASIGMAR1
SCHEMBL6611611 0.91 CCR5 (0.52) LMNACYP2D6MAPTKMT2ASIGMAR1
SCHEMBL6614322 0.91 CCR5 (0.52) LMNACYP2D6MAPTKMT2ASIGMAR1
SCHEMBL6612781 0.89 LMNA (0.53) LMNACYP2D6CHRM2ADRA2ATSHR
SCHEMBL6615053 0.88 OPRL1 (0.55) CHRM2SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL6612028 0.87 LMNA (0.51) LMNACYP2D6CHRM2ADRA2ATSHR
SCHEMBL6611036 0.85 CCR5 (0.52) LMNACYP2D6CHRM2ADRA2ATSHR
SCHEMBL6614791 0.84 OPRM1 (0.42) LMNACYP2D6MAPTKMT2AL3MBTL1
SCHEMBL6613037 0.84 SIGMAR1 (0.49) LMNACYP2D6CHRM2ADRA2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed