SCHEMBL6617622

SCHEMBL6617622

COc1ccc(S(=O)(=O)[C@@](O)(COCc2ccccc2)[C@](N)(Cc2ccccc2)NC(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 11/20 0.50
MMP9 P14780 9/20 0.50
MMP13 P45452 8/20 0.50
MMP2 P08253 6/20 0.44
MMP3 P08254 5/20 0.44
PTPRB P23467 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
ALDH1A1 P00352 3/20 0.40
POLB P06746 1/20 0.38
MMP7 P09237 1/20 0.38
MMP8 P22894 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559637 0.71 MMP13 (0.72) MMP1MMP9MMP13MMP2MMP3
SCHEMBL5771968 0.70 MMP1 (0.44) MMP1MMP9MMP13MMP2MMP3
SCHEMBL8139629 0.70 ALDH1A1 (0.49) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6932195 0.69 MMP13 (0.63) MMP1MMP9MMP13MMP2MMP3
SCHEMBL8843503 0.69 MMP1 (0.52) MMP1MMP9MMP13MMP2MMP3
SCHEMBL8713231 0.69 MMP1 (0.73) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6930656 0.68 MMP1 (0.77) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6929880 0.68 MMP1 (0.76) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6928874 0.67 MMP1 (1.00) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6928756 0.67 MMP13 (0.57) MMP1MMP9MMP13MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086076-B1 SULFONAMIDE INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMA (US) 2004-12-22 EP disclosed