SCHEMBL6624602

SCHEMBL6624602

O=C(O)N(c1ccc(C(F)(F)F)c(OCC(F)(F)F)c1)[N+](=O)[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.36
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPK1 P28482 1/20 0.35
MPI P34949 1/20 0.35
PHOSPHO1 Q8TCT1 1/20 0.35
MRGPRX4 Q96LA9 2/20 0.35
NPSR1 Q6W5P4 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
S1PR2 O95136 1/20 0.34
S1PR4 O95977 1/20 0.34
GAA P10253 1/20 0.34
XBP1 P17861 1/20 0.34
KMT2A Q03164 1/20 0.34
PAX8 Q06710 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
S1PR3 Q99500 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7113987 0.85 RXRA (0.35) RXRALMNAALDH1A1MPIPHOSPHO1
SCHEMBL6607454 0.78 KMO (0.39) LMNAMAPTHTTALDH1A1MAPK1
SCHEMBL17336848 0.78 MAPT (0.36) LMNAMAPTHTTALDH1A1MAPK1
SCHEMBL9836534 0.73 MRGPRX4 (0.39) LMNAMAPTHTTALDH1A1MRGPRX4
SCHEMBL5558208 0.72 RBP4 (0.36)
SCHEMBL312800 0.71 L3MBTL1 (0.53) RXRAALDH1A1MRGPRX4KDM4EHNF4A
SCHEMBL6623841 0.69 RXRA (0.37) RXRALMNAMAPTALDH1A1KDM4E
SCHEMBL21497160 0.67 CYP1A2 (0.49) LMNAMAPTHTTALDH1A1MAPK1
SCHEMBL311898 0.67 KIF11 (0.48) RXRAMAPTHTTALDH1A1KDM4E
SCHEMBL30309512 0.66 ALDH1A1 (0.50) RXRAMAPTHTTALDH1A1MPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379511-A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083652-A1 DIHYDRO-BENZO [b] [1, 4] DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed