SCHEMBL6633355

SCHEMBL6633355

O=Cc1ccc(OCC(=O)OCc2ccccc2)c(C=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
KDM4E B2RXH2 3/20 0.52
MAPT P10636 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
PTGDR2 Q9Y5Y4 2/20 0.47
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
L3MBTL1 Q9Y468 3/20 0.44
MAPK1 P28482 2/20 0.44
POLB P06746 2/20 0.43
LMNA P02545 2/20 0.43
USP2 O75604 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CYP2C9 P11712 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
AKR1B10 O60218 2/20 0.40
AKR1B1 P15121 2/20 0.40
ABCB1 P08183 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28484291 0.85 ALDH1A1 (0.58) ALDH1A1KDM4EMAPTPOLBNPC1
SCHEMBL31312392 0.83 MAOA (0.58) ALDH1A1KDM4EMAPTKMT2AMAOA
SCHEMBL5098548 0.81 NPC1 (0.52) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL6131789 0.80 KDM4E (0.60) ALDH1A1KDM4EMAPTL3MBTL1MAPK1
SCHEMBL7285185 0.80 POLB (0.53) ALDH1A1KDM4EMAPTMAOAMAOB
SCHEMBL7294269 0.80 LMNA (0.54) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL29460406 0.79 MAOA (0.69) ALDH1A1KDM4EMEN1KMT2AMAOA
SCHEMBL22214975 0.79 MAOA (0.69) ALDH1A1KDM4EMEN1KMT2AMAOA
SCHEMBL7284355 0.79 MAOA (0.52) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL2743836 0.79 LMNA (0.50) ALDH1A1KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1079821-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2001-08-29 EP claimed
EP-1079821-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-03-07 EP claimed
WO-1999059570-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-11-25 WO claimed
EP-1067894-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-09-08 EP disclosed
US-6518267-B1 Protease inhibitors SMITHKLINE BEECHAM CORPORATION 2003-02-11 US disclosed
EP-1079821-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2001-08-29 EP disclosed
EP-1079821-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-03-07 EP disclosed
EP-1067894-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-01-17 EP disclosed
WO-1999059570-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-11-25 WO disclosed
WO-1999059526-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-11-25 WO disclosed