SCHEMBL6661590

SCHEMBL6661590

COC(=O)[C@H](Cc1cccs1)NC(C)=O

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.50
CYP2C19 P33261 1/20 0.49
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
CNR2 P34972 1/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
NPC1 O15118 3/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 1/20 0.43
CTSC P53634 2/20 0.43
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PKM P14618 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6661586 1.00 RAB9A (0.50) RAB9ACYP2C19CTSSCTSKCNR2
SCHEMBL25721680 0.86 RAB9A (0.54) RAB9ACYP2C19CTSSCTSKL3MBTL1
SCHEMBL7362447 0.85 CYP2C19 (0.60) RAB9ACYP2C19CTSSCTSKL3MBTL1
SCHEMBL7362451 0.85 CYP2C19 (0.60) RAB9ACYP2C19CTSSCTSKL3MBTL1
SCHEMBL16684110 0.85 CYP2C19 (0.51) RAB9ACYP2C19CTSSCTSKCNR2
SCHEMBL14164208 0.82 CTSK (0.68) RAB9ACYP2C19CTSSCTSKCNR2
SCHEMBL13350918 0.82 RAB9A (0.50) RAB9ACYP2C19CTSSCTSKL3MBTL1
SCHEMBL19051490 0.80 HDAC6 (0.53) HDAC1HDAC6NPC1
SCHEMBL9727077 0.80 CYP2C19 (0.66) RAB9ACYP2C19L3MBTL1NPC1LMNA
SCHEMBL14861287 0.79 HDAC6 (0.70) HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1030854-B1 CATALYSTS FOR ASYMMETRIC SYNTHESIS CONTAINING RIGID CHIRAL LIGANDS PENN STATE RES FOUND (US) 2004-08-18 EP disclosed
US-6380416-B2 CHIRAL BIDENTATE PHOSPHINE LIGANDS WITH CYCLIC RINGS TO RESTRICT CONFORMATIONAL FLEXIBILITY OF THE LIGANDS TO ENHANCE EFFICIENCY; STEREOSELECTIVE HYDROGENATION OF KETONES TO ALCOHOLS, AND A-ACETOAMIDOCINNAMIC ACID TO ACYLAMINO ACIDS THE PENN STATE RESEARCH FOUNDATION 2002-04-30 US disclosed
US-20010047113-A1 Chiral bidentate phosphine ligands with cyclic rings to restrict conformational flexibility of the ligands to enhance efficiency; stereoselective hydrogenation of ketones to alcohols, and a-acetoamidocinnamic acid to acylamino acids THE PENN STATE RESEARCH FOUNDATION 2001-11-29 US disclosed
US-6278024-B1 AS CATALYSTS FOR ASSYMETRIC SYNTHESIS THE PENN STATE RESEARCH FOUNDATION 2001-08-21 US disclosed
US-6207868-B1 BASED ON CHIRAL BIDENTATE PHOSPHINE LIGANDS WITH CYCLIC RING STRUCTURES TO RESTRICT CONFORMATIONAL FLEXIBILITY, ASYMMETRIC SYNTHESIS OF ALCOHOLS BY ENANTIOSELECTIVE HYDROGENATION OF KETONES CATALYZED BY THE CHIRAL LIGANDS THE PENN STATE RESEARCH FOUNDATION 2001-03-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010047113-A1 Chiral bidentate phosphine ligands with cyclic rings to restrict conformational flexibility of the ligands to enhance efficiency; stereoselective hydrogenation of ketones to alcohols, and a-acetoamidocinnamic acid to acylamino acids ADH1A, AASDHPPT, AADAT RAB9A 3780/4885CYP2C19 2761/4885CTSS 3653/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.