SCHEMBL6664555

SCHEMBL6664555

O=C(O)c1ccc2c(c1)C(=O)C(CCc1ccc(Cl)cc1)C(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.40
TP53 P04637 2/20 0.39
MDM2 Q00987 2/20 0.39
DAO P14920 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665845 0.88 CCKBR (0.41) CCKBR
SCHEMBL6685148 0.79 TSHR (0.43) CCKBR
SCHEMBL6678743 0.78 RXRA (0.43) CCKBR
SCHEMBL6681850 0.77 HDAC2 (0.42)
SCHEMBL6683144 0.77 MEN1 (0.43)
SCHEMBL6684713 0.76 TRPV1 (0.37) CCKBR
SCHEMBL6665661 0.76 ALDH1A1 (0.51) TP53
SCHEMBL6665695 0.71 NR4A2 (0.43)
SCHEMBL6684559 0.70 MAPT (0.53) TP53
SCHEMBL6831723 0.70 ALDH1A1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed