SCHEMBL6678743

SCHEMBL6678743

O=C(O)c1ccc2c(c1)C(=O)C(Cc1cccc(Cl)c1)C(=O)N2

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
PDE5A O76074 1/20 0.42
NR4A2 P43354 1/20 0.42
CCKAR P32238 1/20 0.41
CCKBR P32239 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
TAS2R14 Q9NYV8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6683144 0.88 MEN1 (0.43)
SCHEMBL6665845 0.87 CCKBR (0.41) CCKBR
SCHEMBL6665695 0.86 NR4A2 (0.43) NR4A2HCAR2TAS2R14
SCHEMBL6685148 0.85 TSHR (0.43) CCKBR
SCHEMBL6666007 0.84 TRPV1 (0.39)
SCHEMBL6681850 0.83 HDAC2 (0.42)
SCHEMBL6684713 0.82 TRPV1 (0.37) CCKBR
SCHEMBL6668041 0.79 MAPT (0.51)
SCHEMBL6664555 0.78 CCKBR (0.40) CCKBR
SCHEMBL6835347 0.77 RXRA (0.40) RXRARXRBRXRGPDE5ANR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors HICKS JAMES LESTER (US) 2004-03-04 US disclosed
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors MMP13, MMP26, MMP9 RXRA 1763/4885RXRB 1654/4885RXRG 1771/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.