SCHEMBL6685148

SCHEMBL6685148

O=C(O)c1ccc2c(c1)C(=O)C(Cc1ccc(Cl)c(Cl)c1)C(=O)N2

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
CCKBR P32239 1/20 0.42
PYGL P06737 1/20 0.39
PYGM P11217 1/20 0.39
EPHX2 P34913 1/20 0.39
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666007 0.90 TRPV1 (0.39)
SCHEMBL6684713 0.90 TRPV1 (0.37) CCKBR
SCHEMBL6665845 0.88 CCKBR (0.41) CCKBR
SCHEMBL6678743 0.85 RXRA (0.43) CCKBR
SCHEMBL6683144 0.84 MEN1 (0.43)
SCHEMBL6681850 0.84 HDAC2 (0.42) TSHR
SCHEMBL6678534 0.82 MAPT (0.48) EPHX2MAOB
SCHEMBL6665695 0.81 NR4A2 (0.43)
SCHEMBL6664618 0.80 ALDH1A1 (0.53) EPHX2
SCHEMBL6664555 0.79 CCKBR (0.40) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors HICKS JAMES LESTER (US) 2004-03-04 US disclosed
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors MMP13, MMP26, MMP9 TSHR 3050/4885CCKBR 4177/4885PYGL 2691/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.