SCHEMBL6683144

SCHEMBL6683144

O=C(O)c1ccc2c(c1)C(=O)C(Cc1ccccc1)C(=O)N2

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
TTR P02766 1/20 0.41
GFER P55789 1/20 0.40
PTPRC P08575 2/20 0.40
PDPK1 O15530 1/20 0.40
JAK3 P52333 1/20 0.40
TLK2 Q86UE8 1/20 0.40
GSK3B P49841 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ATM Q13315 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PARK7 Q99497 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665845 0.89 CCKBR (0.41)
SCHEMBL6678743 0.88 RXRA (0.43)
SCHEMBL6665695 0.88 NR4A2 (0.43) KMT2A
SCHEMBL6680173 0.86 ALDH1A1 (0.53) MEN1HPGDKMT2APOLBSMN1; SMN2
SCHEMBL6685148 0.84 TSHR (0.43)
SCHEMBL6681850 0.84 HDAC2 (0.42) L3MBTL1POLBSMN1; SMN2
SCHEMBL6684713 0.81 TRPV1 (0.37)
SCHEMBL6664555 0.77 CCKBR (0.40)
SCHEMBL6665661 0.74 ALDH1A1 (0.51) MEN1HPGDKMT2APOLBSMN1; SMN2
SCHEMBL38657178 0.74 GSK3B (0.68) GSK3BL3MBTL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors HICKS JAMES LESTER (US) 2004-03-04 US disclosed
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040043985-A1 6,6-Fused heteroaryl derivatives as matrix metalloproteinase inhibitors MMP13, MMP26, MMP9 MEN1 3612/4885HPGD 564/4885KMT2A 2806/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.