SCHEMBL6665535

SCHEMBL6665535

COc1cc(C(N)=O)ccn1.O=C(O)c1ccc2c(c1)C(=O)CC(=O)N2Cc1ccc(F)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 2/20 0.41
KDM5B Q9UGL1 2/20 0.41
PRKAG1 P54619 2/20 0.41
PRKAA2 P54646 2/20 0.41
PRKAB1 Q9Y478 2/20 0.41
HTR1A P08908 3/20 0.38
GRM2 Q14416 2/20 0.38
ADRA1A P35348 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
PDPK1 O15530 1/20 0.36
CTRB1 P17538 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
GPR52 Q9Y2T5 1/20 0.35
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6668468 0.94 KDM5A (0.41) KDM5AKDM5BPRKAG1PRKAA2PRKAB1
SCHEMBL6665674 0.92 P2RX3 (0.40) KDM5AKDM5BPRKAG1PRKAA2PRKAB1
SCHEMBL6669305 0.90 PRKAG1 (0.41) KDM5AKDM5BPRKAG1PRKAA2PRKAB1
SCHEMBL6666674 0.88 KDM4C (0.42) KDM5AKDM5BGRM2OPRK1KCNH2
SCHEMBL6666692 0.87 PRKAG1 (0.45) KDM5AKDM5BPRKAG1PRKAA2PRKAB1
SCHEMBL6668559 0.84 NNMT (0.41) KDM5AKDM5BPRKAG1PRKAA2PRKAB1
SCHEMBL6665427 0.83 NNMT (0.43) PRKAG1PRKAA2PRKAB1GRM2OPRK1
SCHEMBL6664538 0.81 NNMT (0.45) PRKAG1PRKAA2PRKAB1OPRK1KCNH2
SCHEMBL6663006 0.81 PRKAG1 (0.40) KDM5AKDM5BPRKAG1PRKAA2PRKAB1
SCHEMBL6668051 0.79 PTGDR2 (0.43) PRKAG1PRKAA2PRKAB1OPRK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed