SCHEMBL6668051

SCHEMBL6668051

COc1ccc(C(N)=O)cn1.O=C(O)c1ccc2c(c1)C(=O)CC(=O)N2Cc1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.43
NNMT P40261 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
TP53 P04637 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CPT2 P23786 1/20 0.40
CPT1A P50416 1/20 0.40
CPT1B Q92523 1/20 0.40
OPRM1 P35372 4/20 0.40
OPRK1 P41145 4/20 0.39
PRKAG1 P54619 2/20 0.39
PRKAA2 P54646 2/20 0.39
PRKAB1 Q9Y478 2/20 0.39
KCNH2 Q12809 1/20 0.39
OPRD1 P41143 3/20 0.39
MEN1 O00255 1/20 0.38
CASP6 P55212 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664538 0.93 NNMT (0.45) PTGDR2NNMTOPRM1OPRK1PRKAG1
SCHEMBL6665722 0.90 NNMT (0.43) NNMTMAOBOPRM1OPRK1KCNH2
SCHEMBL6669305 0.90 PRKAG1 (0.41) PTGDR2NNMTOPRM1OPRK1PRKAG1
SCHEMBL6665427 0.89 NNMT (0.43) PTGDR2NNMTOPRM1OPRK1PRKAG1
SCHEMBL6668559 0.88 NNMT (0.41) PTGDR2NNMTOPRM1OPRK1PRKAG1
SCHEMBL6665669 0.84 CPT2 (0.43) PTGDR2TP53SMN1; SMN2CPT2CPT1A
SCHEMBL6665674 0.82 P2RX3 (0.40) PTGDR2OPRK1PRKAG1PRKAA2PRKAB1
SCHEMBL6666674 0.80 KDM4C (0.42) MAOBSMN1; SMN2OPRK1KCNH2MEN1
SCHEMBL6665535 0.79 KDM5A (0.41) PTGDR2OPRK1PRKAG1PRKAA2PRKAB1
SCHEMBL6665423 0.79 NNMT (0.41) NNMTMAOAMAOBOPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed