SCHEMBL6663006

SCHEMBL6663006

NC(=O)c1ccncc1.O=C(O)c1ccc2c(c1)C(=O)CC(=O)N2Cc1ccc(Cl)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAG1 P54619 4/20 0.40
PRKAB1 Q9Y478 4/20 0.40
PRKAA2 P54646 3/20 0.40
KDM5A P29375 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
CTRB1 P17538 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HPGD P15428 1/20 0.37
PTGER4 P35408 1/20 0.37
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.35
PRKAA1 Q13131 1/20 0.35
GPR52 Q9Y2T5 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666692 0.93 PRKAG1 (0.45) PRKAG1PRKAB1PRKAA2KDM5AKDM5B
SCHEMBL6664683 0.92 KMT2A (0.43) PRKAG1PRKAB1PRKAA2CTRB1MEN1
SCHEMBL6667091 0.92 CTRB1 (0.39) PRKAG1PRKAB1PRKAA2KDM5AKDM5B
SCHEMBL6670369 0.89 PRKAG1 (0.43) PRKAG1PRKAB1PRKAA2CTRB1MEN1
SCHEMBL6668468 0.87 KDM5A (0.41) PRKAG1PRKAB1PRKAA2KDM5AKDM5B
SCHEMBL6663894 0.86 ALDH1A1 (0.45) PRKAG1PRKAB1PRKAA2KDM5AKDM5B
SCHEMBL6665669 0.86 CPT2 (0.43) PRKAG1PRKAB1PRKAA2MEN1KMT2A
SCHEMBL6668559 0.84 NNMT (0.41) PRKAG1PRKAB1PRKAA2KDM5AKDM5B
SCHEMBL6667930 0.81 KMT2A (0.51) PRKAG1PRKAB1PRKAA2MEN1KMT2A
SCHEMBL6665535 0.81 KDM5A (0.41) PRKAG1PRKAB1PRKAA2KDM5AKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed