SCHEMBL6664538

SCHEMBL6664538

COc1ccc(C(N)=O)cn1.O=C(O)c1ccc2c(c1)C(=O)CC(=O)N2Cc1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.45
SCN9A Q15858 1/20 0.42
ABCB1 P08183 1/20 0.40
OPRM1 P35372 4/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
P2RX3 P56373 3/20 0.39
OPRK1 P41145 4/20 0.39
PRKAG1 P54619 3/20 0.39
PRKAA2 P54646 3/20 0.39
PRKAB1 Q9Y478 3/20 0.39
KCNH2 Q12809 1/20 0.39
OPRD1 P41143 3/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6668051 0.93 PTGDR2 (0.43) NNMTABCB1OPRM1PTGDR2OPRK1
SCHEMBL6669305 0.92 PRKAG1 (0.41) NNMTSCN9AABCB1OPRM1PTGDR2
SCHEMBL6665427 0.91 NNMT (0.43) NNMTABCB1OPRM1PTGDR2OPRK1
SCHEMBL6668559 0.90 NNMT (0.41) NNMTABCB1OPRM1PTGDR2OPRK1
SCHEMBL6665674 0.89 P2RX3 (0.40) PTGDR2P2RX3OPRK1PRKAG1PRKAA2
SCHEMBL6665722 0.87 NNMT (0.43) NNMTOPRM1OPRK1KCNH2OPRD1
SCHEMBL6670369 0.83 PRKAG1 (0.43) PTGDR2PRKAG1PRKAA2PRKAB1
SCHEMBL6665535 0.81 KDM5A (0.41) PTGDR2OPRK1PRKAG1PRKAA2PRKAB1
SCHEMBL6668468 0.80 KDM5A (0.41) PTGDR2OPRK1PRKAG1PRKAA2PRKAB1
SCHEMBL6665581 0.78 NNMT (0.43) NNMTSCN9AABCB1OPRM1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed