SCHEMBL6667472

SCHEMBL6667472

O=C(NCCc1ccc(Cl)cc1)c1n[nH]c2c(NC3CCOCC3)cc(CN3CCOCC3)cc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
INSR P06213 1/20 0.41
IGF1R P08069 1/20 0.41
ALK Q9UM73 1/20 0.41
KDM4E B2RXH2 1/20 0.41
KCNH2 Q12809 6/20 0.41
POLA1 P09884 2/20 0.41
CHRM1 P11229 2/20 0.41
HTR2A P28223 2/20 0.41
MCHR1 Q99705 2/20 0.41
MAPT P10636 1/20 0.41
ENPP2 Q13822 3/20 0.40
GSK3B P49841 1/20 0.40
CYP2D6 P10635 1/20 0.40
AKR1C3 P42330 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6667470 0.84 INSR (0.39) RAB9AINSRIGF1RALKKCNH2
SCHEMBL6667762 0.83 MEN1 (0.42) MEN1GAARAB9AKMT2AKDM4E
SCHEMBL6667777 0.82 RAB9A (0.55) MEN1GAARAB9AKMT2AKDM4E
SCHEMBL6666561 0.80 MAPT (0.39) MEN1GAARAB9AKMT2AKDM4E
SCHEMBL6669289 0.79 NPC1 (0.40) MEN1GAARAB9AKMT2AKDM4E
SCHEMBL6695646 0.78 POLA1 (0.54) MEN1KMT2AKCNH2POLA1ENPP2
SCHEMBL6974853 0.77 KCNH2 (0.47) RAB9AKCNH2POLA1ENPP2GSK3B
SCHEMBL6666496 0.76 BACE1 (0.38) MEN1GAARAB9AKMT2AKDM4E
SCHEMBL6980565 0.74 KCNH2 (0.44) KCNH2POLA1ENPP2
SCHEMBL6666113 0.74 RAB9A (0.47) MEN1GAARAB9AKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004019940-A1 METHOD OF PREVENTING OR TREATING ATHEROSCLEROSIS OR RESTENOSIS PHARMACIA & UPJOHN COMPANY (US) 2004-03-11 WO claimed
WO-2004019940-A1 METHOD OF PREVENTING OR TREATING ATHEROSCLEROSIS OR RESTENOSIS PHARMACIA & UPJOHN COMPANY (US) 2004-03-11 WO disclosed