SCHEMBL6669289

SCHEMBL6669289

CN(Cc1cc(CN2CCOCC2)cc2c(=O)c(C(=O)NCCc3ccc(Cl)cc3)n[nH]c12)CC1CCCO1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
KDM4E B2RXH2 1/20 0.38
MRGPRX1 Q96LB2 1/20 0.37
KCNH2 Q12809 4/20 0.36
POLA1 P09884 2/20 0.36
BACE1 P56817 1/20 0.36
MCHR1 Q99705 3/20 0.36
CYP2D6 P10635 2/20 0.36
CHRM1 P11229 2/20 0.36
HTR2A P28223 2/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
ENPP2 Q13822 1/20 0.36
HTR3A P46098 1/20 0.36
MAPT P10636 1/20 0.36
EGFR P00533 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6699726 0.81 POLA1 (0.48) KDM4EKCNH2POLA1CYP2D6MEN1
SCHEMBL6667762 0.81 MEN1 (0.42) KDM4EKCNH2POLA1BACE1MCHR1
SCHEMBL6667472 0.79 MEN1 (0.41) KDM4EKCNH2POLA1MCHR1CYP2D6
SCHEMBL6667777 0.76 RAB9A (0.55) NPC1KDM4EKCNH2BACE1MCHR1
SCHEMBL6666496 0.76 BACE1 (0.38) KDM4EKCNH2POLA1BACE1MCHR1
SCHEMBL6974853 0.76 KCNH2 (0.47) NPC1KCNH2POLA1RAB9AENPP2
SCHEMBL6980565 0.74 KCNH2 (0.44) KCNH2POLA1ENPP2
SCHEMBL6669285 0.74 POLA1 (0.35) NPC1KDM4EKCNH2POLA1RAB9A
SCHEMBL6666561 0.71 MAPT (0.39) KDM4EKCNH2POLA1MEN1GAA
SCHEMBL6667754 0.71 AKR1C3 (0.39) NPC1KCNH2POLA1RAB9AENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004019940-A1 METHOD OF PREVENTING OR TREATING ATHEROSCLEROSIS OR RESTENOSIS PHARMACIA & UPJOHN COMPANY (US) 2004-03-11 WO claimed