SCHEMBL6667909

SCHEMBL6667909

CN1C(=O)C(Cc2ccc(F)c(Cl)c2)C(=O)c2cc(C(=O)O)ccc21.COc1ccc(C(N)=O)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.40
KDM5A P29375 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
MAPK1 P28482 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
OPRK1 P41145 4/20 0.34
KCNH2 Q12809 1/20 0.34
ABCB1 P08183 1/20 0.34
P2RX3 P56373 2/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
SCD O00767 1/20 0.33
OPRM1 P35372 3/20 0.33
HTR1A P08908 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665581 0.91 NNMT (0.43) NNMTMKNK1MKNK2OPRK1KCNH2
SCHEMBL6665423 0.89 NNMT (0.41) NNMTKDM5AKDM5BMKNK1MKNK2
SCHEMBL6663534 0.88 NNMT (0.41) NNMTKDM5AKDM5BMKNK1MKNK2
SCHEMBL6681227 0.86 PRKAG1 (0.39) KDM5AKDM5B
SCHEMBL6664479 0.86 ROCK2 (0.40) KDM5AKDM5BPSEN1PSEN2APH1B
SCHEMBL6669268 0.79 ROCK2 (0.38) KDM5AKDM5BPSEN1PSEN2APH1B
SCHEMBL6669305 0.79 PRKAG1 (0.41) NNMTKDM5AKDM5BOPRK1KCNH2
SCHEMBL6685279 0.79 NR1H2 (0.38) KDM5AKDM5B
Niacinamide SCHEMBL6669309 0.79 PSEN1 (0.41) MKNK1MKNK2PSEN1PSEN2APH1B
SCHEMBL6680077 0.78 NR1H2 (0.40) KDM5AKDM5BPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed