SCHEMBL6665581

SCHEMBL6665581

CN1C(=O)C(Cc2ccc(Cl)cc2)C(=O)c2cc(C(=O)O)ccc21.COc1ccc(C(N)=O)cn1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.43
P2RX3 P56373 4/20 0.38
SCN9A Q15858 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
ROCK2 O75116 3/20 0.37
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
OPRK1 P41145 4/20 0.36
KCNH2 Q12809 1/20 0.36
ABCB1 P08183 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
OPRM1 P35372 3/20 0.34
NTRK1 P04629 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6667909 0.91 NNMT (0.40) NNMTP2RX3MKNK1MKNK2OPRK1
SCHEMBL6665423 0.91 NNMT (0.41) NNMTMKNK1MKNK2OPRK1KCNH2
SCHEMBL6663534 0.86 NNMT (0.41) NNMTMKNK1MKNK2OPRK1KCNH2
SCHEMBL6664550 0.85 ROCK2 (0.43) MRGPRX4ROCK2OPRK1
SCHEMBL6663962 0.84 ROCK2 (0.46) ROCK2
SCHEMBL6664538 0.78 NNMT (0.45) NNMTP2RX3SCN9AMRGPRX4MKNK1
SCHEMBL6664479 0.76 ROCK2 (0.40) ROCK2
SCHEMBL6678968 0.76 NR1H2 (0.49)
SCHEMBL6665597 0.75 ROCK2 (0.41) ROCK2OPRK1
SCHEMBL6662847 0.75 TSHR (0.41) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed