SCHEMBL6663534

SCHEMBL6663534

CN1C(=O)C(Cc2cccc(F)c2)C(=O)c2cc(C(=O)O)ccc21.COc1ccc(C(N)=O)cn1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NNMT P40261 2/20 0.41
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
MAOB P27338 1/20 0.37
PARP10 Q53GL7 1/20 0.37
OPRK1 P41145 2/20 0.36
KCNH2 Q12809 1/20 0.36
GRM5 P41594 1/20 0.35
NR4A2 P43354 2/20 0.35
HPGDS O60760 1/20 0.35
KDM5A P29375 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
OPRM1 P35372 2/20 0.34
OPRD1 P41143 2/20 0.34
CCKBR P32239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665423 0.91 NNMT (0.41) NNMTMKNK1MKNK2MAOBOPRK1
SCHEMBL6664526 0.88 PARP10 (0.44) MAOBPARP10NR4A2CCKBR
SCHEMBL6667909 0.88 NNMT (0.40) NNMTMKNK1MKNK2MAOBOPRK1
SCHEMBL6665581 0.86 NNMT (0.43) NNMTMKNK1MKNK2MAOBOPRK1
SCHEMBL6664500 0.85 NR1H2 (0.41) NR4A2KDM5AKDM5BCCKBR
SCHEMBL6662371 0.85 MAOB (0.38) MAOBPARP10OPRK1NR4A2KDM5A
Niacinamide SCHEMBL6669309 0.76 PSEN1 (0.41) MKNK1MKNK2
SCHEMBL6669379 0.76 NNMT (0.43) NNMTMKNK1MKNK2MAOBHPGDS
SCHEMBL6678968 0.76 NR1H2 (0.49) CCKBR
SCHEMBL6665597 0.75 ROCK2 (0.41) OPRK1KDM5AKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014388-A1 6,6-FUSED HETEROARYL DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed