SCHEMBL6667543

SCHEMBL6667543

Cc1oc2ccc(NC(=O)C3CCC3)nc2c1CCN(C)Cc1ccc2ccncc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1F P30939 1/20 0.44
GSK3B P49841 2/20 0.39
ABL1 P00519 9/20 0.35
MAP4K1 Q92918 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
PRMT3 O60678 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HSP90AA1 P07900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550329 0.87 KDM4E (0.40) GSK3BABL1ALDH1A1PRMT3
SCHEMBL6672030 0.79 HTR1F (0.46) HTR1FALDH1A1TSHRCYP1A2CYP2D6
SCHEMBL8191020 0.76 HTR1F (0.42) HTR1FALDH1A1KMT2APRMT3MAPT
SCHEMBL8546411 0.75 ROCK2 (0.37) CYP1A2KMT2APRMT3NPC1RAB9A
SCHEMBL6669755 0.74 HTR1F (0.45) HTR1FGSK3BALDH1A1TSHRCYP1A2
SCHEMBL8548082 0.70 MKNK1 (0.38)
SCHEMBL6668295 0.69 HTR1F (0.44) HTR1FALDH1A1KMT2ANPC1RAB9A
SCHEMBL8551238 0.69 ROCK1 (0.37) ALDH1A1PRMT3RAB9AMAPT
SCHEMBL8550195 0.68 MEN1 (0.44) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8553305 0.67 SMN1; SMN2 (0.42) ALDH1A1TSHRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696439-B1 HETEROCYCLIC IMINES SUCH AS 2-METHYL-3-(2-(N',N'-DIETHYLAMINO) ETHYL)-5-(4-PROPANESULFONYLBENZAMIDE)FURO(3,2-B)PYRIDINE, HYDROCHLORIDE, USED AS SEROTONIN RECEPTOR ANTAGONISTS FOR PROPHYLAXIS OF HEADACHES ELI LILLY AND COMPANY 2004-02-24 US disclosed
EP-1155020-B1 FURO[3,2-B]PYRIDINES AS 5-HT1F AGONISTS LILLY CO ELI (US) 2004-02-04 EP disclosed