SCHEMBL6672827

SCHEMBL6672827

CCOC(=O)CC[C@@H]1Cc2ccccc2C12CCNCC2

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.43
SIGMAR1 Q99720 3/20 0.41
KCNH2 Q12809 1/20 0.40
GRIN2B Q13224 1/20 0.40
NOTUM Q6P988 1/20 0.38
NAMPT P43490 1/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6669828 0.82 HTR2A (0.36) OPRM1SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL6668923 0.81 HTR2A (0.35) SIGMAR1
SCHEMBL6669198 0.75 SIGMAR1 (0.38) SIGMAR1
SCHEMBL6672759 0.73 DRD2 (0.46)
SCHEMBL6670052 0.72 SIGMAR1 (0.38) SIGMAR1
SCHEMBL10531104 0.71 NOTUM (0.48) NOTUMNAMPTCYP4F2CYP4A11
SCHEMBL6672242 0.71 AKT1 (0.40)
SCHEMBL6672515 0.71 AKT1 (0.40)
SCHEMBL14529886 0.69 OPRM1 (0.45) OPRM1SIGMAR1
SCHEMBL6670168 0.68 DRD2 (0.38) OPRM1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399432-A1 SPIROPIPERIDINE COMPOUNDS AS LIGANDS FOR ORL-1 RECEPTOR PFIZER INC. (US) 2004-03-24 EP disclosed
WO-2003000677-A1 SPIROPIPERIDINE COMPOUNDS AS LIGANDS FOR ORL-1 RECEPTOR PFIZER PHARMACEUTICALS INC. (JP) 2003-01-03 WO disclosed