SCHEMBL6674607

SCHEMBL6674607

O=C(NCc1ccc(-c2ccccc2)cc1)Oc1ccc([N+](=O)[O-])s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATG4B Q9Y4P1 3/20 0.55
ALDH1A1 P00352 4/20 0.51
CASP3 P42574 4/20 0.51
SENP8 Q96LD8 4/20 0.51
SENP7 Q9BQF6 4/20 0.51
SENP6 Q9GZR1 4/20 0.51
L3MBTL1 Q9Y468 4/20 0.51
POLB P06746 3/20 0.51
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
CDK2 P24941 1/20 0.45
GSK3A P49840 1/20 0.45
GSK3B P49841 1/20 0.45
DYRK1A Q13627 1/20 0.45
HIPK4 Q8NE63 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
ADAMTS5 Q9UNA0 1/20 0.44
LMNA P02545 1/20 0.44
EPHX1 P07099 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7038371 0.80 CASP3 (0.59) ATG4BALDH1A1CASP3SENP8SENP7
SCHEMBL6676799 0.80 HDAC1 (0.50) ALDH1A1MEN1KMT2ALMNAEPHX1
SCHEMBL5227781 0.72 MAPT (0.40) ALDH1A1CASP3SENP8SENP7SENP6
SCHEMBL10133046 0.71 MGLL (0.65) ALDH1A1MEN1KMT2ALMNAEPHX1
SCHEMBL3757985 0.71 CYP2C9 (0.60) ALDH1A1MEN1MAPTKMT2AADAMTS5
SCHEMBL28570074 0.71 POLB (0.57) ALDH1A1POLBMEN1KMT2ANPC1
SCHEMBL18541826 0.71 ATG4B (1.00) ATG4BCDK2GSK3AGSK3BDYRK1A
SCHEMBL18529258 0.69 ATG4B (0.64) ATG4BALDH1A1CASP3SENP8SENP7
SCHEMBL599832 0.69 CYP2C9 (0.67) MEN1KMT2AADAMTS5MGLLNPC1
SCHEMBL3274691 0.69 FAAH (0.64) ALDH1A1POLBKMT2AADAMTS5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465613-A2 COMBINATION OF MTP INHIBITORS OR APOB SECRETION INHIBITORS WITH FIBRATES FOR USE AS DRUGS Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2004-10-13 EP disclosed
WO-2003057205-A2 COMBINATION OF MTP INHIBITORS OR APOB SECRETION INHIBITORS WITH FIBRATES FOR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-07-17 WO disclosed
WO-2003004020-A1 HETEROARYL CARBOXYLIC ACID AMIDES, THE PRODUCTION THEREOF AND THE USE OF THE SAME AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-01-16 WO disclosed