SCHEMBL6685637

SCHEMBL6685637

NC(=O)C1(C[CH]C(=O)NCCNc2ccc(OC(F)(F)F)cc2)CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.41
CTSS P25774 8/20 0.40
CTSL P07711 6/20 0.40
EPHX2 P34913 3/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.38
EPHX1 P07099 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686841 0.85 CTSK (0.40) CTSKPOLB
SCHEMBL5404868 0.85 CTSK (0.36) CTSKCTSSKMT2AEPHX1
SCHEMBL5843360 0.76 CTSS (0.53) CTSKCTSSCTSLEPHX2POLB
SCHEMBL5520748 0.72 CYP3A4 (0.47) EPHX2EPHX1
SCHEMBL5842740 0.71 HTT (0.34)
SCHEMBL6685642 0.68 CTSS (0.54) CTSKCTSSCTSLEPHX2POLB
SCHEMBL6686917 0.68 CTSS (0.54) CTSKCTSSCTSLEPHX2POLB
SCHEMBL3021858 0.68 EPHX2 (0.57) EPHX2POLBKMT2ACA12CA1
SCHEMBL9780251 0.67 EPHX2 (0.56) EPHX2POLBKMT2ACA12CA1
SCHEMBL5841440 0.66 CTSS (0.64) CTSKCTSSCTSLPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084842-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed