SCHEMBL6686636

SCHEMBL6686636

COc1ccc(NCCN(C)C(=O)[CH]CC(C)(C)C(N)=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.42
GAA P10253 3/20 0.42
RAB9A P51151 3/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
FFAR1 O14842 1/20 0.37
ALDH1A1 P00352 3/20 0.36
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HIF1A Q16665 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 2/20 0.35
TP53 P04637 1/20 0.35
ESR2 Q92731 1/20 0.35
NOX1 Q9Y5S8 1/20 0.35
CA12 O43570 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6688710 0.89 POLB (0.43) MAPTGAARAB9AMEN1KMT2A
SCHEMBL6687560 0.88 MAPT (0.38) MAPTGAAMAPK1ALDH1A1MEN1
SCHEMBL6689081 0.83 TOP2B (0.36) CA12CA1CA2CA9
SCHEMBL6687217 0.78 PARP1 (0.42) MEN1KMT2A
SCHEMBL4800097 0.73 CTSK (0.42) MAPTGAARAB9AMAPK1HSD17B10
SCHEMBL10798884 0.68 GAA (0.70) MAPTGAARAB9AMAPK1HSD17B10
SCHEMBL29939726 0.68 MAPT (0.59) MAPTGAARAB9AFFAR1ALDH1A1
SCHEMBL5404160 0.67 EPHX2 (0.46) MAPTGAARAB9AALDH1A1NPC1
SCHEMBL5409955 0.66 EPHX2 (0.47) MAPTGAARAB9AALDH1A1NPC1
SCHEMBL9372673 0.66 MAPT (0.52) MAPTGAARAB9AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed