SCHEMBL6689081

SCHEMBL6689081

CN(CCNc1ccc(S(C)(=O)=O)cc1)C(=O)[CH]CC(C)(C)C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TOP2B Q02880 2/20 0.36
TGM2 P21980 1/20 0.35
GSR P00390 2/20 0.34
GHSR Q92847 3/20 0.34
CA1 P00915 6/20 0.33
CA2 P00918 6/20 0.33
CA9 Q16790 3/20 0.33
CA12 O43570 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686636 0.83 MAPT (0.42) CA1CA2CA9CA12
SCHEMBL6688710 0.81 POLB (0.43) CA1CA2CA12
SCHEMBL6687560 0.81 MAPT (0.38)
SCHEMBL6687217 0.77 PARP1 (0.42)
SCHEMBL4799004 0.73 TGM2 (0.38) TGM2GHSRCA1CA2CA9
SCHEMBL13589541 0.70 GSR (0.50) TOP2BGSRGHSRCA1CA2
SCHEMBL6690542 0.67 RORC (0.41) GHSRCA2
SCHEMBL14624916 0.65 CA12 (0.49) TGM2GSRCA1CA2CA9
SCHEMBL13589540 0.64 CA1 (0.45) TGM2GHSRCA1CA2CA9
SCHEMBL8212136 0.64 GHSR (0.47) TGM2GHSRCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed