SCHEMBL6692480

SCHEMBL6692480

CC(C)(C)OC(=O)N[C@H](C(O)CCc1ncc(CCCO)s1)C(Cc1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 5/20 0.38
ADRB1 P08588 5/20 0.38
ADRB3 P13945 5/20 0.38
ATM Q13315 1/20 0.38
KLK5 Q9Y337 2/20 0.37
CTSS P25774 2/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSK P43235 1/20 0.36
PTPRB P23467 1/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 4/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
XBP1 P17861 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664868 0.93 CTSK (0.41) ATMKLK5CTSKALDH1A1
SCHEMBL6663482 0.93 KLK5 (0.41) ATMKLK5CTSSCTSLCTSB
SCHEMBL6666961 0.92 ALDH1A1 (0.39) ATMKLK5CTSSCTSLCTSB
SCHEMBL6668504 0.92 ALDH1A1 (0.39) ATMKLK5CTSSCTSLCTSB
SCHEMBL6666632 0.91 ALDH1A1 (0.40) ATMKLK5CTSSCTSLCTSB
SCHEMBL9378904 0.86 CTSS (0.41) ATMKLK5CTSSCTSLCTSB
SCHEMBL9379291 0.85 ATM (0.39) ATMKLK5CTSSCTSLCTSB
SCHEMBL9373974 0.85 PTPRB (0.39) ATMKLK5CTSSCTSLCTSB
SCHEMBL9372986 0.84 ATM (0.38) ATMKLK5CTSSCTSLCTSB
SCHEMBL9373933 0.84 CTSK (0.39) ATMKLK5CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450795-A1 PEPTIDE ISOSTERES CONTAINING A HETEROCYCLE USEFUL IN THE TREATMENT OF ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2004-09-01 EP claimed
WO-2003047576-A1 PEPTIDE ISOSTERES CONTAINING A HETEROCYCLE USEFUL IN THE TREATMENT OF ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2003-06-12 WO claimed