SCHEMBL9372986

SCHEMBL9372986

CCC(=O)c1cnc(CC[C@H](O)[C@@H](NC(=O)OC(C)(C)C)C(Cc2ccccc2)c2ccccc2)s1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.38
KLK5 Q9Y337 3/20 0.38
CTSK P43235 6/20 0.37
CTSS P25774 3/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
PTPRB P23467 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ACE P12821 1/20 0.36
AKT1 P31749 1/20 0.35
APP P05067 1/20 0.35
REN P00797 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9373974 0.91 PTPRB (0.39) ATMKLK5CTSKCTSSCTSL
SCHEMBL9379291 0.91 ATM (0.39) ATMKLK5CTSKCTSSCTSL
SCHEMBL6666632 0.88 ALDH1A1 (0.40) ATMKLK5CTSKCTSSCTSL
SCHEMBL6666961 0.87 ALDH1A1 (0.39) ATMKLK5CTSKCTSSCTSL
SCHEMBL6668504 0.87 ALDH1A1 (0.39) ATMKLK5CTSKCTSSCTSL
SCHEMBL9378904 0.87 CTSS (0.41) ATMKLK5CTSKCTSSCTSL
SCHEMBL9373933 0.87 CTSK (0.39) ATMKLK5CTSKCTSSCTSL
SCHEMBL6663482 0.86 KLK5 (0.41) ATMKLK5CTSKCTSSCTSL
SCHEMBL6664868 0.86 CTSK (0.41) ATMKLK5CTSKALDH1A1REN
SCHEMBL6692480 0.84 ADRB2 (0.38) ATMKLK5CTSKCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0603309-A1 PEPTIDE ISOTERS CONTAINING A HETEROCYCLE AS H.I.V. INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-06-29 EP disclosed