SCHEMBL6664868

SCHEMBL6664868

CCCCc1cnc(CC[C@H](O)[C@@H](NC(=O)OC(C)(C)C)C(Cc2ccccc2)c2ccccc2)s1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.41
ALDH1A1 P00352 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK5 Q00535 1/20 0.38
ATM Q13315 1/20 0.38
GLS O94925 2/20 0.37
KLK5 Q9Y337 1/20 0.37
REN P00797 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666961 0.95 ALDH1A1 (0.39) CTSKALDH1A1ATMKLK5
SCHEMBL6668504 0.95 ALDH1A1 (0.39) CTSKALDH1A1ATMKLK5
SCHEMBL6692480 0.93 ADRB2 (0.38) CTSKALDH1A1ATMKLK5
SCHEMBL6666632 0.93 ALDH1A1 (0.40) CTSKALDH1A1CCNE1CDK2CDK5
SCHEMBL6663482 0.91 KLK5 (0.41) CTSKALDH1A1ATMKLK5
SCHEMBL9378904 0.86 CTSS (0.41) CTSKATMKLK5
SCHEMBL9372986 0.86 ATM (0.38) CTSKALDH1A1ATMKLK5REN
SCHEMBL9373933 0.86 CTSK (0.39) CTSKALDH1A1ATMKLK5
SCHEMBL9373974 0.85 PTPRB (0.39) CTSKALDH1A1ATMKLK5REN
SCHEMBL9379291 0.85 ATM (0.39) CTSKALDH1A1ATMKLK5REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450795-A1 PEPTIDE ISOSTERES CONTAINING A HETEROCYCLE USEFUL IN THE TREATMENT OF ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2004-09-01 EP disclosed
WO-2003047576-A1 PEPTIDE ISOSTERES CONTAINING A HETEROCYCLE USEFUL IN THE TREATMENT OF ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2003-06-12 WO disclosed