SCHEMBL6693365

SCHEMBL6693365

COc1ccc(C(=O)NC(c2ccccc2)c2c[nH]nc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.59
CYP3A4 P08684 1/20 0.59
GAA P10253 2/20 0.53
LMNA P02545 2/20 0.51
TP53 P04637 2/20 0.51
ADORA1 P30542 1/20 0.47
UTS2R Q9UKP6 3/20 0.46
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
HPGDS O60760 1/20 0.45
TRPA1 O75762 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.43
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43
AURKA O14965 2/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28476592 0.76 ALDH1A1 (0.86) ALDH1A1CYP3A4GAALMNATP53
SCHEMBL28466269 0.72 HPGDS (0.72) ALDH1A1CYP3A4GAALMNAKMT2A
SCHEMBL2008486 0.70 SLC6A9 (0.82) ALDH1A1CYP3A4GAAKMT2AMEN1
SCHEMBL6678578 0.70 MAPT (0.42) ALDH1A1CYP3A4GAALMNAKMT2A
SCHEMBL6689991 0.69 MAPT (0.41) ALDH1A1CYP3A4GAALMNAKMT2A
SCHEMBL3107205 0.69 HPGDS (0.67) ALDH1A1CYP3A4GAALMNAKMT2A
SCHEMBL30530178 0.68 SLC6A9 (0.71) ALDH1A1CYP3A4GAALMNAUTS2R
SCHEMBL6691606 0.68 HSD17B2 (0.41) ALDH1A1CYP3A4GAALMNAKMT2A
SCHEMBL13498069 0.67 LMNA (1.00) LMNATP53KMT2AMEN1HSP90AA1
SCHEMBL28466273 0.67 SLC6A9 (0.68) GAALMNAUTS2RKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043951-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS CAREX S.A. (FR) 2004-05-27 WO claimed