SCHEMBL7098488

SCHEMBL7098488

c1cncc(Cn2cc(-c3ccco3)cn2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.57
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
ADORA3 P0DMS8 1/20 0.45
ADORA2B P29275 1/20 0.45
ALDH1A1 P00352 6/20 0.43
PKM P14618 3/20 0.43
KDM4E B2RXH2 4/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CLK4 Q9HAZ1 1/20 0.42
KDM5B Q9UGL1 1/20 0.42
SCD5 Q86SK9 3/20 0.42
HSD17B10 Q99714 2/20 0.42
SCD O00767 2/20 0.42
HPGD P15428 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
ABL1 P00519 1/20 0.41
BCR P11274 1/20 0.41
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004006 0.86 L3MBTL1 (0.64) L3MBTL1ADORA2AADORA1ALDH1A1KDM4E
SCHEMBL6690784 0.79 ADORA2A (0.50) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7096885 0.79 ADORA2A (0.52) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7097845 0.79 ADORA2A (0.43) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6693887 0.76 MEN1 (0.60) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL6691423 0.75 ADORA2A (0.48) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7096746 0.74 ADORA2A (0.54) ADORA2AADORA1ADORA3ADORA2BALDH1A1
SCHEMBL12068737 0.73 L3MBTL1 (0.56) L3MBTL1ALDH1A1PKMKDM4EKDM5B
SCHEMBL7096791 0.73 ADORA2A (0.48) L3MBTL1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7092539 0.73 ADORA2A (0.50) L3MBTL1ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed