SCHEMBL7096885

SCHEMBL7096885

Nc1cccc(Cn2cc(-c3ccco3)cn2)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.52
ADORA1 P30542 6/20 0.52
ADORA3 P0DMS8 1/20 0.47
ADORA2B P29275 1/20 0.47
ALK Q9UM73 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
SCD5 Q86SK9 6/20 0.44
SCD O00767 3/20 0.43
CREBBP Q92793 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PI4KA P42356 1/20 0.40
PIK3CG P48736 1/20 0.40
PI4KB Q9UBF8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690784 0.85 ADORA2A (0.50) ADORA2AADORA1ADORA3ADORA2BL3MBTL1
SCHEMBL7004006 0.84 L3MBTL1 (0.64) ADORA2AADORA1L3MBTL1SCD5SCD
SCHEMBL6693887 0.81 MEN1 (0.60) ADORA2AADORA1ADORA3ADORA2BMEN1
SCHEMBL7096746 0.80 ADORA2A (0.54) ADORA2AADORA1ADORA3ADORA2BALK
SCHEMBL7098488 0.79 L3MBTL1 (0.57) ADORA2AADORA1ADORA3ADORA2BMEN1
SCHEMBL14712472 0.77 MEN1 (0.68) ADORA2AADORA1ALKMEN1KMT2A
SCHEMBL7097845 0.76 ADORA2A (0.43) ADORA2AADORA1ADORA3ADORA2BMEN1
SCHEMBL7092539 0.76 ADORA2A (0.50) ADORA2AADORA1ADORA3ADORA2BL3MBTL1
SCHEMBL6691423 0.76 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BMEN1
SCHEMBL983078 0.74 L3MBTL1 (0.71) ADORA2AADORA1ALKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed