SCHEMBL6696196

SCHEMBL6696196

CC(C)(C)c1ccc(S(=O)(=O)C(CN2CCNc3ccccc3C2)c2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.40
MAPK1 P28482 1/20 0.38
ALDH1A1 P00352 3/20 0.37
HSD11B1 P28845 2/20 0.36
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
SPPL2A Q8TCT8 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
POLB P06746 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
KCNH2 Q12809 1/20 0.34
BRS3 P32247 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6694497 0.87 MEN1 (0.36) MAPK1ALDH1A1POLBDRD2MEN1
SCHEMBL6697273 0.71 MAPK1 (0.57) MAPK1ALDH1A1DRD2MAPTKDM4E
SCHEMBL10280392 0.66 MAPK1 (0.47) MAPK1ALDH1A1
SCHEMBL31332341 0.64 SIGMAR1 (0.54) ALDH1A1DRD3KCNH2MEN1KMT2A
SCHEMBL6701653 0.63 REN (0.35) POLBDRD2DRD3KCNH2HTT
SCHEMBL10241074 0.60 MAPK1 (0.54) MAOAMAPK1ALDH1A1KCNH2
SCHEMBL7005533 0.58 MAPK1 (0.45) MAPK1
SCHEMBL2849413 0.58 MAOA (0.53) MAOAMAPK1DRD2DRD3KCNH2
SCHEMBL19652058 0.58 MAPK1 (0.69) MAPK1MEN1KMT2A
SCHEMBL11661937 0.58 HTR7 (0.50) ALDH1A1POLBKDM4EMMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040009972-A1 Benzodiazepine inhibitors of mitochondial F1F0 ATP hydrolase and methods of inhibiting F1F0 ATP hydrolase BRISTOL-MYERS COMPANY 2004-01-15 US disclosed
WO-2003106628-A2 BENZODIAZEPINE INHIBITORS OF MITOCHONDIAL F1F0 ATP HYDROLASE AND METHODS OF INHIBITING F1F0 ATP HYDROLASE BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009972-A1 Benzodiazepine inhibitors of mitochondial F1F0 ATP hydrolase and methods of inhibiting F1F0 ATP hydrolase MT-ATP6, MT-CO1, ATP5ME MAOA 606/4885MAPK1 4076/4885ALDH1A1 1084/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.