SCHEMBL6701010

SCHEMBL6701010

COC(=O)c1ccc2ccn(Cc3ccc(S(C)(=O)=O)cc3)c(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA4 P22748 2/20 0.46
CA9 Q16790 2/20 0.46
MAPK8 P45983 5/20 0.45
ALDH1A1 P00352 3/20 0.43
MAPK10 P53779 2/20 0.43
LMNA P02545 1/20 0.43
PTGS2 P35354 4/20 0.43
MAPK9 P45984 1/20 0.43
HDAC11 Q96DB2 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179110 0.92 CA1 (0.40) CA1CA2CA4CA9MAPK8
SCHEMBL6167921 0.88 CA1 (0.41) CA1CA2CA4CA9MAPK8
SCHEMBL2115805 0.87 HDAC6 (0.52) HDAC11HDAC8HDAC6HDAC3HDAC4
SCHEMBL2117651 0.85 MMP13 (0.48) MAPK8ALDH1A1MAPK10LMNASMN1; SMN2
SCHEMBL6703278 0.83 MMP13 (0.60) LMNAHDAC11HDAC8HDAC6HDAC3
SCHEMBL9974663 0.83 PTGS2 (0.45) CA1CA2CA4CA9MAPK8
SCHEMBL6703541 0.83 CYP11B1 (0.49) ALDH1A1MAPK10LMNAHDAC11HDAC8
SCHEMBL6168393 0.83 LMNA (0.46) ALDH1A1MAPK10LMNAHDAC11HDAC8
SCHEMBL6697454 0.82 RORC (0.51) ALDH1A1LMNAPOLBNPC1RAB9A
SCHEMBL6697238 0.81 PDPK1 (0.43) ALDH1A1MAPK10LMNAHDAC11HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040044000-A1 Isoquinoline derivatives as matrix metalloproteinase inhibitors BUNKER AMY MAE (US) 2004-03-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040044000-A1 Isoquinoline derivatives as matrix metalloproteinase inhibitors MMP1, MMP13, MMP9 CA1 1576/4885CA2 503/4885CA4 740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.