SCHEMBL6709802

SCHEMBL6709802

COC(=O)c1ccccc1NC(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.67
CYP1A2 P05177 1/20 0.67
CYP2D6 P10635 1/20 0.67
CYP2C19 P33261 1/20 0.67
NPC1 O15118 1/20 0.64
MAPT P10636 4/20 0.64
ALDH1A1 P00352 2/20 0.64
MEN1 O00255 4/20 0.62
KMT2A Q03164 4/20 0.62
POLB P06746 2/20 0.62
KDM4E B2RXH2 2/20 0.62
APOBEC3A P31941 1/20 0.61
APOBEC3G Q9HC16 1/20 0.61
LMNA P02545 2/20 0.61
ABCG2 Q9UNQ0 1/20 0.60
HPGD P15428 1/20 0.60
MAPK10 P53779 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.59
ELANE P08246 1/20 0.58
PRTN3 P24158 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367856 0.87 LMNA (0.70) TSHRNPC1MAPTALDH1A1MEN1
SCHEMBL7316304 0.87 ALDH1A1 (0.57) TSHRCYP1A2CYP2D6CYP2C19NPC1
SCHEMBL7372951 0.86 KMT2A (0.69) NPC1MAPTALDH1A1MEN1KMT2A
SCHEMBL4094329 0.86 KMT2A (0.66) TSHRNPC1MAPTALDH1A1MEN1
SCHEMBL1309081 0.85 SMN1; SMN2 (0.70) NPC1MAPTALDH1A1MEN1KMT2A
SCHEMBL11665959 0.82 TSHR (0.77) TSHRCYP1A2CYP2D6CYP2C19MAPT
SCHEMBL7374064 0.82 MEN1 (0.78) NPC1MAPTALDH1A1MEN1KMT2A
SCHEMBL6716445 0.82 ALDH1A1 (0.60) MAPTALDH1A1MEN1KMT2AKDM4E
SCHEMBL4443911 0.82 ALOX5 (0.63) NPC1MAPTALDH1A1MEN1KMT2A
SCHEMBL9339256 0.81 TSHR (0.76) TSHRCYP1A2CYP2D6CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004022525-A1 AMIDE DERIVATIVES AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 2004-03-18 WO claimed
WO-2004022525-A1 AMIDE DERIVATIVES AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 2004-03-18 WO disclosed
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed