SCHEMBL671609

SCHEMBL671609

CNc1cc(OCC(F)F)c(C(N)=O)cc1N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
XDH P47989 1/20 0.36
MKNK2 Q9HBH9 1/20 0.35
LRRK2 Q5S007 1/20 0.34
PRKCI P41743 1/20 0.34
MAPT P10636 2/20 0.33
TSHR P16473 1/20 0.33
CNR2 P34972 2/20 0.33
NNMT P40261 2/20 0.33
SIRT2 Q8IXJ6 1/20 0.32
GSK3B P49841 1/20 0.32
IKBKB O14920 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.31
HTT P42858 2/20 0.31
LMNA P02545 1/20 0.31
ACACB O00763 1/20 0.31
NTRK1 P04629 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11951408 0.89 PRKCI (0.40) MKNK2PRKCIMAPTTSHRGSK3B
SCHEMBL670579 0.85 ALDH1A1 (0.40) KDM4EALDH1A1GAAMAPTTSHR
SCHEMBL1726279 0.79 PTGES (0.49) KDM4EALDH1A1GAAMAPTHTT
SCHEMBL11951461 0.78 TAS1R3 (0.42) ALDH1A1CNR2
SCHEMBL10170839 0.76 FADS1 (0.51) KDM4EMAPTTSHRHTT
SCHEMBL1725449 0.76 PTGES (0.47) ALDH1A1LRRK2CNR2
SCHEMBL1725448 0.76 PTGES (0.47) ALDH1A1LRRK2CNR2
SCHEMBL27964720 0.74 HTR2A (0.34) ALDH1A1MKNK2LRRK2HTTLMNA
SCHEMBL27147584 0.74 KDM4E (0.49) KDM4EALDH1A1GLAGAAMAPT
SCHEMBL672665 0.74 PTGER4 (0.37) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606036-A1 NEW COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2013-06-26 EP disclosed
CN-103097359-A Novel compounds BOEHRINGER INGELHEIM INT 2013-05-08 CN disclosed
WO-2012022793-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-02-23 WO disclosed
WO-2010100249-A1 3H-IMIDAZO [4, 5 -C] PYRIDINE- 6 -CARBOXAMIDES AS ANTI- INFLAMMATORY AGENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-10 WO disclosed