SCHEMBL6745377

SCHEMBL6745377

CCOC(=O)N1CSC[C@@H]1C(=O)N[C@@H](Cc1ccc(NC(=O)c2ccccc2C(F)(F)F)cc1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 16/20 0.44
ITGB1 P05556 13/20 0.44
FPR2 P25090 1/20 0.39
KCNK3 O14649 1/20 0.39
KCNK9 Q9NPC2 1/20 0.39
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6744943 0.87 ITGA4 (0.50) ITGA4ITGB1
SCHEMBL6745542 0.84 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL6741663 0.84 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL6742360 0.83 ITGB1 (0.46) ITGA4ITGB1FPR2
SCHEMBL6742904 0.83 ITGA4 (0.49) ITGA4ITGB1
SCHEMBL6744273 0.82 ITGA4 (0.52) ITGA4ITGB1
SCHEMBL6741921 0.82 ITGB1 (0.47) ITGA4ITGB1
SCHEMBL6741830 0.81 ITGA4 (0.54) ITGA4ITGB1
SCHEMBL6744349 0.81 FPR2 (0.46) ITGA4ITGB1FPR2
SCHEMBL27563993 0.81 ITGA4 (0.43) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed
CN-1313855-A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta UPJOHN CO (US) 2001-09-19 CN disclosed