SCHEMBL6744637

SCHEMBL6744637

Cc1csc(C2=CCC=C2c2cc(F)c(S(C)(=O)=O)c(F)c2)n1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 4/20 0.33
CASP1 P29466 1/20 0.32
GLA P06280 1/20 0.32
GABRA1 P14867 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
GABRA5 P31644 2/20 0.31
GABRA3 P34903 2/20 0.31
GABRA2 P47869 2/20 0.31
CYP2E1 P05181 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2A6 P11509 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2B6 P20813 1/20 0.31
MIF P14174 1/20 0.30
PPARA Q07869 1/20 0.30
CYP19A1 P11511 1/20 0.30
ADORA2A P29274 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6744707 0.80 HPGD (0.39) CASP1RAB9A
SCHEMBL6746763 0.78 NR1H2 (0.31) TYK2GLAGABRA1GABRG2GABRB3
SCHEMBL6729457 0.78 PTGS2 (0.40) TYK2CASP1GLAGABRA1GABRG2
SCHEMBL6746288 0.77 CASP1 (0.35) CASP1
SCHEMBL6749937 0.75 PTGS2 (0.36) CASP1
SCHEMBL6747157 0.75 TGFBR1 (0.37) CASP1GLACYP2A6
SCHEMBL6730758 0.75 TYK2 (0.33) TYK2CASP1GLA
SCHEMBL6746753 0.74 PTGS2 (0.45) CASP1
SCHEMBL6746730 0.73 PTGS2 (0.38) CASP1
SCHEMBL6728005 0.73 CYP2E1 (0.43) GLAGABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US claimed
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US disclosed