SCHEMBL6765008

SCHEMBL6765008

O=C(OC1Cc2ccccc2OC1c1ccccc1)c1cc(O)c(O)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 1.00
DYRK1A Q13627 8/20 0.89
IGF1R P08069 1/20 0.89
BACE1 P56817 5/20 0.58
BCL2 P10415 4/20 0.58
PSMB5 P28074 4/20 0.58
SNCA P37840 4/20 0.58
PGD P52209 4/20 0.58
MET P08581 3/20 0.58
KDM4E B2RXH2 3/20 0.58
MEN1 O00255 3/20 0.58
MAPT P10636 3/20 0.58
RECQL P46063 3/20 0.58
KMT2A Q03164 3/20 0.58
TDP1 Q9NUW8 3/20 0.58
PKM P14618 3/20 0.58
PKMYT1 Q99640 2/20 0.58
SIRT6 Q8N6T7 2/20 0.58
USP2 O75604 2/20 0.58
CYP3A4 P08684 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20043083 1.00 HSP90AB1 (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL17972588 1.00 HSP90AB1 (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL17220841 1.00 HSP90AB1 (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL17220840 1.00 HSP90AB1 (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL24984288 0.94 DYRK1A (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL30987004 0.94 DYRK1A (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL30141006 0.94 DYRK1A (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL24983851 0.94 DYRK1A (1.00) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL21381204 0.88 HSP90AB1 (0.78) HSP90AB1DYRK1AIGF1RBACE1BCL2
SCHEMBL19319148 0.87 HSP90AB1 (0.77) HSP90AB1DYRK1AIGF1RBACE1BCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11952358-B2 Flavan-3-ol analogs and anti-inflammatory activity HONG KONG BAPTIST UNIVERSITY (CN) 2024-04-09 US disclosed
US-20230159482-A1 FLAVAN-3-OL ANALOGS AND ANTI-INFLAMMATORY ACTIVITY HONG KONG BAPTIST UNIVERSITY (CN) 2023-05-25 US disclosed
CN-111406755-A Camellia nitidissima theaflavin medicament for resisting novel coronavirus and preparation method and application thereof 韶关学院 2020-07-14 CN disclosed
CN-111406755-A Camellia nitidissima theaflavin medicament for resisting novel coronavirus and preparation method and application thereof 韶关学院 2020-07-14 CN disclosed
US-10308624-B2 Catalytic enantioselective synthesis of 2-aryl chromenes and related phosphoramidite ligands and catalyst compounds NORTHWESTERN UNIVERSITY (US) 2019-06-04 US disclosed
US-20180099943-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds NORTHWESTERN UNIVERSITY 2018-04-12 US disclosed
US-9840487-B2 Catalytic enantioselective synthesis of 2-aryl chromenes and related phosphoramidite ligands and catalyst compounds NORTHWESTERN UNIVERSITY (US) 2017-12-12 US disclosed
US-20170217919-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds NORTHWESTERN UNIVERSITY 2017-08-03 US disclosed
US-9624190-B2 Catalytic enantioselective synthesis of 2-aryl chromenes and related phosphoramidite ligands and catalyst compounds NORTHWESTERN UNIVERSITY (US) 2017-04-18 US disclosed
US-20160221982-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds NORTHWESTERN UNIVERSITY 2016-08-04 US disclosed
US-9309217-B2 Catalytic enantioselective synthesis of 2-aryl chromenes and related phosphoramidite ligands and catalyst compounds NORTHWESTERN UNIVERSITY (US) 2016-04-12 US disclosed
US-20150315168-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-11-05 US disclosed
US-6713506-B2 INHIBITING PROTEASOMAL CHYMOTRYPSIN-LIKE ACTIVITY UNIVERSITY OF SOUTH FLORIDA 2004-03-30 US disclosed
US-20020151582-A1 Tea polyphenol esters and analogs thereof for cancer prevention and treatment SOUTH FLORIDA, UNIVERSITY OF 2002-10-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170217919-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds PNP, PPA1, CDS2 HSP90AB1 4603/4885DYRK1A 372/4885IGF1R 1063/4885
US-11952358-B2 Flavan-3-ol analogs and anti-inflammatory activity IL1A, IL6, IL1B HSP90AB1 794/4885DYRK1A 4754/4885IGF1R 1285/4885
US-20160221982-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds PNP, PPA1, CDS2 HSP90AB1 4603/4885DYRK1A 372/4885IGF1R 1063/4885
US-10308624-B2 Catalytic enantioselective synthesis of 2-aryl chromenes and related phosphoramidite ligands and catalyst compounds PNP, PPA1, CDS2 HSP90AB1 4603/4885DYRK1A 372/4885IGF1R 1063/4885
US-20150315168-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds PNP, PPA1, CDS2 HSP90AB1 4603/4885DYRK1A 372/4885IGF1R 1063/4885
US-20230159482-A1 FLAVAN-3-OL ANALOGS AND ANTI-INFLAMMATORY ACTIVITY IL1A, IL6, IL1B HSP90AB1 794/4885DYRK1A 4754/4885IGF1R 1285/4885
US-20020151582-A1 Tea polyphenol esters and analogs thereof for cancer prevention and treatment GCG, CTSG, CTRL HSP90AB1 506/4885DYRK1A 4828/4885IGF1R 4632/4885
US-20180099943-A1 Catalytic Enantioselective Synthesis of 2-Aryl Chromenes and Related Phosphoramidite Ligands and Catalyst Compounds PNP, PPA1, CDS2 HSP90AB1 4603/4885DYRK1A 372/4885IGF1R 1063/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.