SCHEMBL6772068

SCHEMBL6772068

CCCc1nn(-c2ccc(C(C)C)cc2)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
LMNA P02545 1/20 0.57
OPRM1 P35372 10/20 0.53
ALPL P05186 2/20 0.53
NPSR1 Q6W5P4 2/20 0.52
KMT2A Q03164 1/20 0.52
GAA P10253 1/20 0.50
HSP90AB1 P08238 4/20 0.48
HSP90AA1 P07900 2/20 0.42
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479730 0.87 OPRM1 (0.54) ALDH1A1LMNAOPRM1NPSR1GAA
SCHEMBL6767582 0.86 ALDH1A1 (0.56) ALDH1A1LMNAOPRM1ALPLNPSR1
SCHEMBL6163724 0.86 ALDH1A1 (0.65) ALDH1A1LMNAOPRM1ALPLNPSR1
SCHEMBL6770401 0.82 OPRM1 (0.77) ALDH1A1LMNAOPRM1NPSR1HSP90AB1
SCHEMBL6767006 0.82 OPRM1 (0.58) OPRM1HSP90AB1HSP90AA1OPRD1OPRK1
SCHEMBL6770454 0.81 ALDH1A1 (0.48) ALDH1A1LMNAOPRM1ALPLNPSR1
SCHEMBL6772480 0.81 ALDH1A1 (0.67) ALDH1A1LMNAOPRM1ALPLNPSR1
SCHEMBL7533974 0.80 OPRM1 (0.47) ALDH1A1LMNAOPRM1NPSR1KMT2A
SCHEMBL6767198 0.80 L3MBTL1 (0.44) ALDH1A1LMNAALPLNPSR1KMT2A
SCHEMBL6770500 0.79 OPRM1 (0.61) OPRM1HSP90AB1HSP90AA1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed