SCHEMBL6769175

SCHEMBL6769175

CC(C)(C)N(CCOc1cccc2c(N)nccc12)C(=O)OC(=O)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 7/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
CYBB P04839 1/20 0.33
NCF1 P14598 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
HTR1B P28222 1/20 0.32
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
HPGD P15428 2/20 0.32
RAF1 P04049 4/20 0.31
ATM Q13315 1/20 0.31
PDGFRB P09619 1/20 0.31
BRAF P15056 1/20 0.31
PDGFRA P16234 1/20 0.31
KDR P35968 1/20 0.31
MALT1 Q9UDY8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6769172 0.86 L3MBTL1 (0.38) RIPK1NOS3NOS1NOS2CYBB
SCHEMBL6770681 0.82 KLKB1 (0.32) BRAF
SCHEMBL5662541 0.70 SCN9A (0.49) KDM4EALDH1A1HPGDATM
SCHEMBL6770030 0.69 ALDH1A1 (0.48) CYBBNCF1HTR1BKDM4EALDH1A1
Trifluoroacetic Acid SCHEMBL6770678 0.69 F7 (0.33) BRAF
SCHEMBL5663479 0.66 HTR1B (0.58) NOS3NOS1NOS2CYBBNCF1
Hydrochloric Acid SCHEMBL5661310 0.65 HTR1B (0.57) NOS3NOS1NOS2CYBBNCF1
Trifluoroacetic Acid SCHEMBL6768943 0.62 F10 (0.50) KDM4EHPGD
SCHEMBL3468335 0.60 PDK2 (0.40) KDM4EALDH1A1
SCHEMBL873662 0.60 NOS2 (0.59) NOS3NOS1NOS2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825181-B1 ORALLY ADMINISTRATED TO EXHIBIT A STRONG ANTICOAGULANT EFFECT BY INHIBITING ACTIVATED BLOOD- COAGULATION FACTOR X AJINOMOTO CO., INC. (JP) 2004-11-30 US disclosed
EP-1065200-A1 AMINOISOQUINOLINE DERIVATIVES Ajinomoto Co., Inc. (JP) 2001-01-03 EP disclosed