SCHEMBL6772805

SCHEMBL6772805

CCOCc1nc2c(N)nc(C)cc2n1CCCCNC(=O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 7/20 0.44
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
BRD4 O60885 2/20 0.40
HDAC2 Q92769 1/20 0.39
GCGR P47871 1/20 0.39
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MCHR1 Q99705 1/20 0.37
PPARD Q03181 1/20 0.37
HPGD P15428 3/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6768615 0.91 TLR7 (0.39) HDAC3HDAC1TLR8TLR7MCHR1
SCHEMBL6772889 0.90 SMN1; SMN2 (0.48) HDAC3HDAC1NPC1RAB9AHPGD
SCHEMBL6772832 0.89 TP53 (0.47) HDAC3HDAC1BRD4HDAC2TLR8
SCHEMBL6779395 0.88 TLR7 (0.46) HDAC3HDAC1HDAC2TLR8TLR7
SCHEMBL6778818 0.86 HDAC3 (0.47) HDAC3HDAC1HDAC2TLR8TLR7
SCHEMBL6778546 0.85 ALDH1A1 (0.45) HDAC3HDAC1HDAC2TLR8TLR7
SCHEMBL6777494 0.85 DRD2 (0.39) TLR7ALDH1A1
SCHEMBL6768551 0.84 TLR7 (0.42) TRPV1HDAC3HDAC1BRD4HDAC2
SCHEMBL6774530 0.84 TRPV1 (0.42) TRPV1HDAC3HDAC1HDAC2GCGR
SCHEMBL6771963 0.83 MAPT (0.46) NPC1RAB9AMCHR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6720333-B2 IMMUNE RESPONSE MODIFIERS; CYTOKINE BIOSYNTHESIS; VIRAL AND NEOPLASTIC DISEASES; N-(4-(4-AMINO-6,7-DIMETHYL-1H-IMIDAZO (4,5-C)PYRIDIN-1-YL)BUTYL)BENZAMIDE 3M INNOVATIVE PROPERTIES COMPANY 2004-04-13 US claimed