SCHEMBL677469

SCHEMBL677469

[CH2]Cc1ccc(CCCCCCCC)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.63
ADRA2A P08913 2/20 0.63
ADORA3 P0DMS8 2/20 0.63
TACR2 P21452 2/20 0.63
SLC6A2 P23975 2/20 0.63
SLC6A4 P31645 2/20 0.63
SLC6A3 Q01959 2/20 0.63
ALDH1A1 P00352 2/20 0.63
HSD17B10 Q99714 2/20 0.63
KDM4E B2RXH2 1/20 0.63
LMNA P02545 1/20 0.63
SHBG P04278 1/20 0.63
TP53 P04637 1/20 0.63
CYP3A4 P08684 1/20 0.63
HSPD1 P10809 1/20 0.63
ADRB3 P13945 1/20 0.63
HTR2C P28335 1/20 0.63
HSPE1 P61604 1/20 0.63
HIF1A Q16665 1/20 0.63
TST Q16762 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2915276 1.00 ESR1 (0.63) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL9753538 1.00 ESR1 (0.63) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL7530233 1.00 ESR1 (0.63) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL1611473 1.00 ESR1 (0.63) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL698308 1.00 ESR1 (0.63) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL1609476 0.98 ESR1 (0.59) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL363054 0.91 CA2 (0.54) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL23849704 0.88 ESR1 (0.77) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL2511615 0.88 ESR1 (0.77) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL10980557 0.88 ESR1 (0.77) ESR1ADRA2AADORA3TACR2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 153 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116987045-A Heteroatom-containing substituted benzoxazinone derivative and preparation method and application thereof 中国医学科学院药物研究所 2023-11-03 CN claimed
US-20220213210-A1 COMBINATION THERAPY OF MULTIPLE SCLEROSIS COMPRISING A CD20 LIGAND MABION SA (PL) 2022-07-07 US claimed
EP-3720880-A1 COMBINATION THERAPY OF MULTIPLE SCLEROSIS COMPRISING A CD20 LIGAND Mabion SA (PL) 2020-10-14 EP claimed
WO-2019110643-A1 COMBINATION THERAPY OF MULTIPLE SCLEROSIS COMPRISING A CD20 LIGAND MABION SA (PL) 2019-06-13 WO claimed
US-20170312249-A1 MODULATORS OF 14-3-3 FUNCTIONALITY AND USES THEREOF UNIVERSITY OF SOUTH AUSTRALIA (AU) 2017-11-02 US claimed
WO-2016054680-A1 MODULATORS OF 14-3-3 FUNCTIONALITY AND USES THEREOF UNIVERSITY OF SOUTH AUSTRALIA (AU) 2016-04-14 WO claimed
CN-103724215-A Novel derivative of 2-amino-2-[2-(4-octylphenyl)ethyl]-1,3-propandiol and application of novel derivative ZHENJIANG SHENGAN PHARMACEUTICAL CO LTD 2014-04-16 CN claimed
CN-101478961-B S1P receptor modulators for the treatment of multiple sclerosis NOVARTIS AG 2013-11-27 CN claimed
CN-101797241-B Solid pharmaceutical compositions comprising a sip receptor agonist and a sugar alcohol NOVARTIS AG 2013-03-27 CN claimed
CN-101068536-B Dosage regimen of an S1P receptor agonist NOVARTIS AG 2012-12-05 CN claimed
CN-1993115-B Compound formulations of 2-amino-1, 3-propanediol compounds NOVARTIS AG (CH) 2011-12-28 CN claimed
CN-1893934-B Use of sphingosine-1-phosphate (S1P) receptor agonists for the manufacture of a medicament for the treatment of brain degenerative diseases NOVARTIS AG 2010-05-26 CN claimed
CN-101478961-A S1P receptor modulators for the treatment of multiple sclerosis NOVARTIS AG (CH) 2009-07-08 CN claimed
US-20070270499-A1 Use for 2-amino-2-propane-1, 3-diols WELSCH CAROLE 2007-11-22 US claimed
US-20040214897-A1 Uses for 2-amino-2-propane-1,3-diols WELSCH CAROLE 2004-10-28 US claimed
WO-2003009836-A2 NEW USES FOR 2-AMINO-2-PROPANE-1,3-DIOLS NOVARTIS AG (CH) 2003-02-06 WO claimed
WO-1999014204-A1 SUBSTITUTED 1,2,4-TRIAZOLES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY G.D. SEARLE & CO. (US) 1999-03-25 WO claimed
CN-116987045-A Heteroatom-containing substituted benzoxazinone derivative and preparation method and application thereof 中国医学科学院药物研究所 2023-11-03 CN disclosed
US-3957854-A FUEL ADDITIVES, LUBRICANTS THE LUBRIZOL CORPORATION (US) 1976-05-18 US disclosed
US-3957855-A FUEL ADDITIVES, LUBRICANTS THE LUBRIZOL CORPORATION (US) 1976-05-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040214897-A1 Uses for 2-amino-2-propane-1,3-diols DGKB, GLS2, GLS ESR1 2376/4885ADRA2A 720/4885ADORA3 3010/4885
US-20070270499-A1 Use for 2-amino-2-propane-1, 3-diols DGKB, GLS2, GLS ESR1 1805/4885ADRA2A 556/4885ADORA3 2308/4885
US-20170312249-A1 MODULATORS OF 14-3-3 FUNCTIONALITY AND USES THEREOF YWHAH, YWHAG, YWHAB ESR1 4271/4885ADRA2A 4651/4885ADORA3 4060/4885
US-20220213210-A1 COMBINATION THERAPY OF MULTIPLE SCLEROSIS COMPRISING A CD20 LIGAND CD209, MSR1, SIGLEC7 ESR1 2741/4885ADRA2A 1382/4885ADORA3 405/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.