SCHEMBL6775933

SCHEMBL6775933

COc1ccc(Oc2c(C)cc(NC(=O)C(C)C)cc2C)cc1SC(C)C

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 2/20 0.46
KMT2A Q03164 2/20 0.45
THRB P10828 5/20 0.43
THRA P10827 4/20 0.43
MEN1 O00255 1/20 0.41
AR P10275 1/20 0.40
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
RORC P51449 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6769373 0.85 MTNR1B (0.47) MTNR1BTHRBTHRARORC
SCHEMBL6765992 0.85 AR (0.52) KMT2ATHRBTHRAMEN1AR
SCHEMBL6769412 0.74 KDM4E (0.34) MTNR1BTHRBTHRAKDM4ELMNA
SCHEMBL6775732 0.74 RORC (0.54) MTNR1BKMT2ATHRBTHRAMEN1
SCHEMBL6775887 0.73 THRB (0.36) KMT2ATHRBMEN1KDM4ELMNA
SCHEMBL7094647 0.70 THRB (0.61) THRBTHRARORC
SCHEMBL7097286 0.70 THRB (0.75) THRBTHRARORC
SCHEMBL8799875 0.70 THRB (0.60) THRBTHRARORC
SCHEMBL6769171 0.70 THRB (0.31) KMT2ATHRBMEN1RORC
SCHEMBL8798523 0.69 THRB (0.54) THRBTHRARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723717-B1 CARDIAC-SPARING; SIDE EFFECT REDUCTION THE UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER 2004-04-20 US disclosed