SCHEMBL6776140

SCHEMBL6776140

COC(=O)CCN1CCCN(Cc2ccc(Cl)cc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHKA P35790 3/20 0.55
CACNA1G O43497 3/20 0.54
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
TP53 P04637 1/20 0.51
DRD4 P21917 2/20 0.49
CCR2 P41597 2/20 0.49
DRD2 P14416 1/20 0.49
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48
POLB P06746 1/20 0.48
HTR7 P34969 1/20 0.47
CHRM1 P11229 1/20 0.47
HTR2A P28223 1/20 0.47
MCHR1 Q99705 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6776114 0.85 CCR2 (0.58) CHKACCR2
SCHEMBL8571246 0.84 CHKA (0.50) CHKAKDM4EALDH1A1CCR2
SCHEMBL6770035 0.83 KDM4E (0.57) CACNA1GKDM4EALDH1A1DRD4CCR2
SCHEMBL11632873 0.82 ALDH1A1 (0.56) CACNA1GKDM4EALDH1A1TP53DRD4
Hydrochloric Acid SCHEMBL8479099 0.82 KMT2A (0.63) KDM4EALDH1A1MAPTHTR7
SCHEMBL3032788 0.81 NPC1 (0.66) KDM4EALDH1A1TP53HRH3
SCHEMBL13073679 0.80 CACNA1G (0.53) CACNA1GKDM4EALDH1A1DRD4GAA
SCHEMBL5483874 0.79 SMN1; SMN2 (0.61) KDM4EALDH1A1TP53MAPTPOLB
SCHEMBL22639905 0.78 SIGMAR1 (0.61) CACNA1GKDM4EALDH1A1DRD4DRD2
SCHEMBL2056181 0.78 CHKA (0.77) CHKAKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6686353-B1 PREVENTING BLOOD MONOCYTES AND LYMPHOCYTES FROM INFILTRATING TISSUE TEIJIN INTELLECTUAL PROPERTY CENTER LIMITED (JP) 2004-02-03 US disclosed
EP-0914319-B1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LTD (JP) 2001-11-21 EP disclosed
EP-0914319-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1999-05-12 EP disclosed
WO-1997044329-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1997-11-27 WO disclosed