SCHEMBL6776495

SCHEMBL6776495

COc1cc(CCCN2CC3CCCC(C2=O)N3C(=O)OC(C)(C)C)cc(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FKBP5 Q13451 2/20 0.51
FKBP1A P62942 9/20 0.40
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6778877 0.90 FKBP5 (0.51) FKBP5KMT2AHTT
SCHEMBL6778408 0.87 FKBP5 (0.50) FKBP5KMT2AHTT
SCHEMBL6780481 0.86 FKBP5 (0.55) FKBP5FKBP1AKMT2AMEN1
SCHEMBL6775961 0.84 KMT2A (0.42) FKBP5FKBP1AKMT2A
SCHEMBL6785002 0.81 KMT2A (0.41) FKBP5FKBP1AKMT2A
SCHEMBL6778841 0.80 KMT2A (0.41) FKBP5FKBP1AKMT2A
SCHEMBL6785090 0.80 FKBP1A (0.50) FKBP5FKBP1AKMT2AMEN1HTT
SCHEMBL6779072 0.80 FKBP5 (0.54) FKBP5FKBP1AKMT2AHTT
SCHEMBL6779125 0.79 FKBP1A (0.44) FKBP5FKBP1AKMT2AMEN1HTT
SCHEMBL6776517 0.76 FKBP5 (0.45) FKBP5FKBP1AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818643-B1 3,9-DIAZABICYCLO(3.3.1)NONAN-2-ONE DERIVATIVES; PEPTIDYL-PROLYL ISOMERASE (PPIASE OR ROTAMASE) INHIBITORS; NEUROPROTECTIVE AGENTS BRISTOL-MYERS SQUIBB COMPANY 2004-11-16 US disclosed
WO-2001042245-A1 NEUROTROPHIC BICYCLIC DIAMIDES BRISTOL-MYERS SQUIBB COMPANY (US) 2001-06-14 WO disclosed