SCHEMBL6783532

SCHEMBL6783532

COc1ccc(CCCCN2C[C@H]3CC[C@@H](C2=O)N3C(=O)C(F)(F)c2cc(OC)c(OC)c(OC)c2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP5 Q13451 2/20 0.47
FKBP1A P62942 3/20 0.41
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37
TUBB8 Q3ZCM7 1/20 0.37
TUBA3E Q6PEY2 1/20 0.37
TUBA1A Q71U36 1/20 0.37
TUBA1C Q9BQE3 1/20 0.37
TUBB6 Q9BUF5 1/20 0.37
TUBB2B Q9BVA1 1/20 0.37
TUBB1 Q9H4B7 1/20 0.37
ALDH1A1 P00352 5/20 0.37
TDP1 Q9NUW8 2/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6774588 0.97 FKBP5 (0.47) FKBP5FKBP1ATUBB4ATUBBTUBA3C
SCHEMBL6779072 0.93 FKBP5 (0.54) FKBP5FKBP1AALDH1A1TDP1POLB
SCHEMBL6779125 0.92 FKBP1A (0.44) FKBP5FKBP1AMEN1KMT2AHTT
SCHEMBL6776757 0.88 FKBP1A (0.47) FKBP5FKBP1AALDH1A1KMT2AMAPT
SCHEMBL6781032 0.81 FKBP1A (0.47) FKBP5FKBP1AALDH1A1MEN1KMT2A
SCHEMBL6778408 0.77 FKBP5 (0.50) FKBP5ALDH1A1TDP1POLBRECQL
SCHEMBL6784892 0.76 FKBP1A (0.48) FKBP5FKBP1AALDH1A1
SCHEMBL6785000 0.75 FKBP1A (0.45) FKBP5FKBP1AALDH1A1MEN1KMT2A
SCHEMBL6778877 0.74 FKBP5 (0.51) FKBP5ALDH1A1TDP1POLBRECQL
SCHEMBL6785090 0.74 FKBP1A (0.50) FKBP5FKBP1AMEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818643-B1 3,9-DIAZABICYCLO(3.3.1)NONAN-2-ONE DERIVATIVES; PEPTIDYL-PROLYL ISOMERASE (PPIASE OR ROTAMASE) INHIBITORS; NEUROPROTECTIVE AGENTS BRISTOL-MYERS SQUIBB COMPANY 2004-11-16 US disclosed