SCHEMBL6785000

SCHEMBL6785000

COc1cc(C(F)(F)C(=O)N2[C@@H]3CC[C@H]2C(=O)N(C(CCc2ccccc2)CCc2ccccc2)C3)cc(OC)c1OC

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 5/20 0.45
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 4/20 0.38
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
MEN1 O00255 2/20 0.36
G6PD P11413 1/20 0.36
METAP2 P50579 1/20 0.36
MAPT P10636 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
FKBP5 Q13451 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6776757 0.85 FKBP1A (0.47) FKBP1AALDH1A1KMT2AMAPTFKBP5
SCHEMBL6781032 0.82 FKBP1A (0.47) FKBP1AALDH1A1KMT2ALMNAMEN1
SCHEMBL6784892 0.79 FKBP1A (0.48) FKBP1AALDH1A1FKBP5
SCHEMBL6783532 0.75 FKBP5 (0.47) FKBP1AALDH1A1KMT2AMEN1MAPT
SCHEMBL6779072 0.71 FKBP5 (0.54) FKBP1AALDH1A1KMT2AFKBP5
SCHEMBL6780693 0.67 SIGMAR1 (0.42) ALDH1A1KMT2AMEN1SIGMAR1
SCHEMBL6779167 0.66 SIGMAR1 (0.46) FKBP1AALDH1A1SIGMAR1
SCHEMBL6774415 0.61 BCHE (0.39) FKBP1AALDH1A1KMT2AMEN1G6PD
SCHEMBL6628799 0.61 FKBP5 (0.69) FKBP1AALDH1A1FKBP5
SCHEMBL6627612 0.61 FKBP1A (0.57) FKBP1AFKBP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818643-B1 3,9-DIAZABICYCLO(3.3.1)NONAN-2-ONE DERIVATIVES; PEPTIDYL-PROLYL ISOMERASE (PPIASE OR ROTAMASE) INHIBITORS; NEUROPROTECTIVE AGENTS BRISTOL-MYERS SQUIBB COMPANY 2004-11-16 US disclosed