SCHEMBL6784809

SCHEMBL6784809

Cn1ncc(Nc2ccccc2F)c1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 1/20 0.46
TSHR P16473 1/20 0.45
P4HTM Q9NXG6 1/20 0.43
KDM4E B2RXH2 1/20 0.43
RAB9A P51151 4/20 0.42
NPC1 O15118 2/20 0.42
MAPT P10636 1/20 0.42
AURKA O14965 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
MAPK8 P45983 1/20 0.40
BRD4 O60885 1/20 0.40
BPTF Q12830 1/20 0.40
KAT2B Q92831 1/20 0.40
BRD9 Q9H8M2 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
EPHB3 P54753 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6786512 0.82 BPTF (0.48) TSHRKDM4ERAB9AMAPTSMN1; SMN2
SCHEMBL6785353 0.78 BPTF (0.58) KDM4ESMN1; SMN2GAABRD4BPTF
SCHEMBL6784797 0.77 PDE10A (0.56) RAB9ANPC1MAPTSMN1; SMN2GAA
SCHEMBL6786035 0.74 FLT1 (0.56) GAABRD4BPTFKAT2BBRD9
SCHEMBL6786160 0.74 BPTF (0.44) KDM4ERAB9ANPC1MAPTSMN1; SMN2
SCHEMBL6789292 0.72 SMN1; SMN2 (0.48) KDM4ERAB9ANPC1MAPTSMN1; SMN2
SCHEMBL4256425 0.70 FABP4 (0.65) CXCL8KDM4EMAPTMAPK8CYP1A2
SCHEMBL6787123 0.69 BPTF (0.50) RAB9ANPC1MAPTSMN1; SMN2BRD4
SCHEMBL10919213 0.69 HDAC1 (0.41) KDM4EMAPTAURKASMN1; SMN2GAA
SCHEMBL29793294 0.68 CXCL8 (0.55) CXCL8KDM4ERAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6686373-B2 ANALGESICS; ANTIINFLAMMATORY AGENT WARNER-LAMBERT COMPANY LLC 2004-02-03 US disclosed
US-20030130277-A1 Pyrazoloquinolinone derivatives as protein kinase C inhibitors KAWAMURA KIYOSHI (JP) 2003-07-10 US disclosed
EP-1310498-A2 Pyrazoloquinolinone derivatives as protein kinase C inhibitors PFIZER INC. (US) 2003-05-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030130277-A1 Pyrazoloquinolinone derivatives as protein kinase C inhibitors PRKCB, PRKCA, PRKCG CXCL8 1528/4885TSHR 3713/4885P4HTM 2516/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.